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DiscoveryProbe™ Protease Inhibitor Library
130个蛋白酶抑制剂的独特集合,用于高通量筛选(HTS)和高含量筛选(HCS)。

DiscoveryProbe™ Protease Inhibitor Library

产品编号:L1035
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Sample solution is provided at 25 µL, 10mM.

Click and Customize the Panel with your own choices of compounds/size/qtuanties/chemical forms etc.

引用文献

1. Huang L, Li L, et al. "Targeting HIV-1 Protease Autoprocessing for High-throughput Drug Discovery and Drug Resistance Assessment." Sci Rep. 2019 Jan 22;9(1):301. PMID:30670786

HTS Facility Partners

质量控制

相关生物数据

CA-074 Me

相关生物数据

CA-074 Me

相关生物数据

Semagacestat (LY450139)

相关生物数据

Semagacestat (LY450139)

相关生物数据

PAC-1

相关生物数据

PAC-1

相关生物数据

DiscoveryProbe™ Protease Inhibitor Library

Signaling Pathway

Bcl-2 Family Research Area
Bcl-2 Family Compare Products
p53 Research Area
p53 Compare Products

Featured Products of the Library

Catalog No. Product Name Summary Targets CAS Number Smiles
A2576 E-64 Cysteine protease inhibitor,irriversible Cathepsin 66701-25-5 CC(C)CC(C(=O)NCCCCN=C(N)N)NC(=O)C1C(O1)C(=O)O
A2606 Epoxomicin Proteasome inhibitor Proteasome 134381-21-8 CCC(C)C(C(=O)NC(C(C)O)C(=O)NC(CC(C)C)C(=O)C1(CO1)C)NC(=O)C(C(C)CC)N(C)C(=O)C
A4018 YO-01027 (Dibenzazepine, DBZ) γ-secretase inhibitor Gamma Secretase 209984-56-5 CC(C(=O)NC1C2=CC=CC=C2C3=CC=CC=C3N(C1=O)C)NC(=O)CC4=CC(=CC(=C4)F)F
A4054 17-AAG (KOS953) Hsp90 inhibitor HSP 75747-14-7 CC1CC(C(C(C=C(C(C(C=CC=C(C(=O)NC2=CC(=O)C(=C(C1)C2=O)NCC=C)C)OC)OC(=O)N)C)C)O)OC
A8200 DAPT (GSI-IX) γ-secretase inhibitor,potent and specific Amyloid β 208255-80-5 CC(C(=O)NC(C1=CC=CC=C1)C(=O)OC(C)(C)C)NC(=O)CC2=CC(=CC(=C2)F)F
A8203 Ritonavir HIV protease inhibitor HIV Protease 155213-67-5 CC(C)C1=NC(=CS1)CN(C)C(=O)NC(C(C)C)C(=O)NC(CC2=CC=CC=C2)CC(C(CC3=CC=CC=C3)NC(=O)OCC4=CN=CS4)O
A8206 Darunavir HIV-1 protease inhibitor HIV Protease 635728-49-3 CCO.CC(C)CN(CC(C(CC1=CC=CC=C1)NC(=O)OC2COC3C2CCO3)O)S(=O)(=O)C4=CC=C(C=C4)N
A8239 CA-074 Me Cathepsin B inhibitor Cathepsin 147859-80-1 CCCNC(=O)C1C(O1)C(=O)NC(C(C)CC)C(=O)N2CCCC2C(=O)OC
Download the Protease-Inhibitor-Library - XLSX       Download the Protease-Inhibitor-Library - SDF

Advantages

  • Available in stock with overnight delivery and free shipping over $500
  • Cost-effective and competitive price to save your findings
  • Potent, selective and cell-permeable in inhibiting or activating target molecules
  • Diverse in chemical structure and route of administration (oral/i.m/i.v injection etc.)
  • Detailed files describing potency, selectivity and applications etc.
  • Supported by published data from top peer-reviewed journals
  • Guaranteed high quality with NMR and HPLC validation

Storage and Shipping Information

Form Pre-dissolved DMSO solutions Stability -20°C: 3 months
-80°C: 6 months
Packaging 96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode.
General tips For obtaining a higher solubility , please warm the tube at 37°C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.
Shipping Condition Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request

Compound Library Composition